Osaka Medical and Pharmaceutical University · Graduate School of Pharmaceutical Sciences / Department of Pharmacy / Faculty of Pharmaceutical Sciences · 教授

Research keywords機能性分子・有機化学・多元素創薬化学・医薬化学・ケミカルバイオロジー・ケミカルスペース・VDRリガンド・アンドロゲン受容体拮抗薬

This is a public-data preview. Personalized fit, contact angles, and saved workflows require sign-in.

• Design, synthesis and structural development of nonsecosteroidal VDR ligands based on the C,C′-diphenyl-m-carborane scaffold2026 · European Journal of Medicinal Chemistry / Elsevier BV / 302
• Structure-activity relationship and crystallographic analyses of non-secosteroidal vitamin D receptor ligands bearing diphenylsilane core as a hydrophobic pharmacophore2025 · Bioorg. Med. Chem. / Elsevier BV / 128
• Modular synthesis of unsymmetrical 1,1’-disubstituted ferrocenes by sequential Suzuki-Miyaura cross-coupling of 1,1’-diborylferrocene2025 · Chemistry - Eur. J. / in press
• Physicochemical characterization of B-hydroxyphenyl phosphine borane derivatives and their evaluation as nuclear estrogen receptor ligands2024 · RSC Med. Chem. / Royal Society of Chemistry (RSC) / 15 / 1

• リンを用いた新しい分子設計手法の開発と医薬リード化合物の創製2023
• 有機金属化合物の特性を利用した分子設計法の開発と医薬リード創出2023
• ホスフィンボラン構造を用いた新規ケミカルスペースの開拓と生物活性化合物の創出法の提案2020
• 細胞増殖シグナル制御化合物と受容体の分子間相互作用の解明2020

• Official profile