Ryugaku Jinja · Professor Archive
Public Professor Archive
Yoshiaki Isobe磯部 義明
Shiga University of Medical Science · Unclassified · 特任教授
Shiga University of Medical Science · Unclassified · 特任教授
This is a public-data preview. Personalized fit, contact angles, and saved workflows require sign-in.
- N-(6-phenylpyridazin-3-yl)benzenesulfonamides as highly potent, brain-permeable, and orally active kynurenine monooxygenase inhibitors2021 · Bioorganic & Medicinal Chemistry Letters, 2021年02月01日, 査読有り
- Identification of 2-fluoro-8-methyl-11-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)-5H-dibenzo[b,e][1,4]diazepine with clozapine-like mixed activities at muscarinic acetylcholine, dopamine, and serotonin receptors2021 · Bioorganic & Medicinal Chemistry Letters, 2021年05月15日, 査読有り
- Discovery of N-(6-(5-fluoro-2-(piperidin-1-yl)phenyl)pyridazin-3-yl)-1-(tetrahydro-2H-pyran-4-yl)methanesulfonamide as a brain-permeable and metabolically stable kynurenine monooxygenase inhibitor2021 · Bioorganic & Medicinal Chemistry Letters, 2021年07月15日, 査読有り
- Synthesis and pharmacological evaluation of 11-(1,6-dimethyl-1,2,3,6-tetrahydropyridin-4-yl)-5H-dibenzo[b,e][1,4]diazepines with clozapine-like receptor occupancy at dopamine D1/D2 receptor2020 · Bioorganic & Medicinal Chemistry Letters, 2020年03月01日, 査読有り
Next stepSign in for fit and contact guidance
Personalized fit, contact angles, and saved workflows require sign-in.